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primary ovarian insufficiency/obésité

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17-acetamido-4-azasteroid derivatives as androgen receptor modulators

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FIELD OF THE INVENTION The present invention relates to 17-acetamido-4-azasteroid derivatives, their synthesis, and their use as androgen receptor modulators. More particularly, the compounds of the present invention are tissue-selective androgen receptor modulators (SARMs) and are thereby useful

Fluorinated 4-azasteroids as androgen receptor modulators

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FIELD OF THE INVENTION The present invention relates to fluorinated 4-azasteroid derivatives, their synthesis, and their use as androgen receptor modulators. More particularly, the compounds of the present invention are tissue-selective androgen receptor modulators (SARMs) and are thereby useful for

N-(2-benzyl)-2-phenylbutanamides as androgen receptor modulators

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FIELD OF THE INVENTION The present invention relates to N-(2-benzyl)-2-phenylbutanamide derivatives, their synthesis, and their use as androgen receptor modulators. More particularly, the compounds of the present invention are tissue-selective androgen receptor modulators (SARMs) and are thereby

Androgen receptor modulators

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FIELD OF THE INVENTION The present invention relates to 3-4 fused-imidazolyl steroidal derivatives, their synthesis, and their use as androgen receptor modulators. More particularly, the compounds of the present invention are tissue-selective androgen receptor modulators (SARMs) and are thereby

N-(2-benzyl)-2-phenylbutanamides as androgen receptor modulators

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FIELD OF THE INVENTION The present invention relates to N-(2-benzyl)-2-phenylbutanamide derivatives, their synthesis, and their use as androgen receptor modulators. More particularly, the compounds of the present invention are tissue-selective androgen receptor modulators (SARMs) and are thereby

17-Heterocyclic-4-azasteroid derivatives as androgen receptor modulators

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FIELD OF THE INVENTION The present invention relates to 17-heterocyclic-4-azasteroid derivatives, their synthesis, and their use as androgen receptor modulators. More particularly, the compounds of the present invention are tissue-selective androgen receptor modulators (SARMs) and are thereby useful

Polymorphs of an androgen receptor modulator

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FIELD OF THE INVENTION The present invention relates to crystalline and amorphous forms and solvates of N-(3H-imidazo[4,5-B]pyridin-2-ylmethyl)-2-fluoro-4-methyl-3-oxo-4-aza-5-a- lpha-androst-1-en-17-beta-carboxamide, a tissue-selective androgen receptor modulator (SARM). This SARM is thereby useful

N-(2-benzyl)-2-phenylbutanamides as androgen receptor modulators

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FIELD OF THE INVENTION The present invention relates to N-(2-benzyl)-2-phenylbutanamide derivatives, their synthesis, and their use as androgen receptor modulators. More particularly, the compounds of the present invention are tissue-selective androgen receptor modulators (SARMs) and are thereby

Fluorinated 4-azasteroid derivatives as androgen receptor modulators

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FIELD OF THE INVENTION The present invention relates to fluorinated 4-azasteroid derivatives, their synthesis, and their use as androgen receptor modulators. More particularly, the compounds of the present invention are tissue-selective androgen receptor modulators and are thereby useful for the

4-azasteroid derivatives as androgen receptor modulators

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FIELD OF THE INVENTION The present invention relates to 4-azasteroid derivatives, their synthesis, and their use as androgen receptor modulators. More particularly, the compounds of the present invention are tissue-selective androgen receptor modulators and are thereby useful for the treatment of

Fluorinated 4-azasteroid derivatives as androgen receptor modulators

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FIELD OF THE INVENTION The present invention relates to fluorinated 4-azasteroid derivatives, their synthesis, and their use as androgen receptor modulators. More particularly, the compounds of the present invention are tissue-selective androgen receptor modulators and are thereby useful for the

21-Heterocyclic-4-azasteroid derivatives as androgen receptor modulators

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FIELD OF THE INVENTION The present invention relates to 21-benzimidazole-4-azasteroid and 21-azabenzimidazole-azasteroid derivatives, their synthesis, and their use as androgen receptor modulators. More particularly, the compounds of the present invention are tissue-selective androgen receptor

17-Acetamido-4-azasteroid derivatives as androgen receptor modulators

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FIELD OF THE INVENTION The present invention relates to 17-acetamido-4-azasteroid derivatives, their synthesis, and their use as androgen receptor modulators. More particularly, the compounds of the present invention are tissue-selective androgen receptor modulators (SARMs) and are thereby useful

17-heterocyclic-4-azasteroid derivatives as androgen receptor modulators

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FIELD OF THE INNENTION The present invention relates to 17-heterocyclic-4-azasteroid derivatives, their synthesis, and their use as androgen receptor modulators. More particularly, the compounds of the present invention are tissue-selective androgen receptor modulators and are thereby useful for the

17-acetamido-4-azasteroid derivatives as androgen receptor modulators

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FIELD OF THE EVICTION The present invention relates to 17-acetamido-4-azasteroid derivatives, their synthesis, and their use as androgen receptor modulators. More particularly, the compounds of the present invention are tissue-selective androgen receptor modulators (SARMs) and are thereby useful for
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