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Bioorganic and Medicinal Chemistry Letters 2013-Nov

Bicyclic and tricyclic heterocycle derivatives as histamine H3 receptor antagonists for the treatment of obesity.

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Manuel de Lera Ruiz
Junying Zheng
Michael Y Berlin
Kevin D McCormick
Robert G Aslanian
Robert West
Joyce Hwa
Jean Lachowicz
Margaret van Heek

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Abstrè

A novel series of non-imidazole bicyclic and tricyclic histamine H3 receptor antagonists has been discovered. Compound 17 was identified as a centrally penetrant molecule with high receptor occupancy which demonstrates robust oral activity in rodent models of obesity. In addition compound 17 possesses clean CYP and hERG profiles and shows no behavioral changes in the Irwin test.

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