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antidiarrheals/infarction

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Comparison of stably expressed rat UGT1.1 and UGT2B1 in the glucuronidation of opioid compounds.

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Opioids are important drugs used as analgesics, antitussives, antidiarrheals, and in the therapy of myocardial infarctions, and as antagonists of opioid intoxication. The glucuronidation of these compounds, catalyzed by UDP-glucuronosyltransferases (UGTs), is well known to be a primary step in their
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