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acetamide/obesitas

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Diazepane acetamide derivatives as selective 11B-HSD1 inhibitors

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FIELD OF THE INVENTION The present invention relates to diazepane-acetamide derivatives as selective inhibitors of the enzyme 11-beta-hydroxysteroid dehydrogenase type 1 (11.beta.-HSD-1) and the use of such compounds for the treatment and prevention of metabolic syndrome, diabetes, insulin

Diazepane-acetamide derivatives as selective 11.beta.-HSD1 inhibitors

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FIELD OF THE INVENTION The present invention relates to diazepane-acetamide derivatives as selective inhibitors of the enzyme 11-beta-hydroxysteroid dehydrogenase type 1 (11.beta.-HSD-1) and the use of such compounds for the treatment and prevention of metabolic syndrome, diabetes, insulin

4-substituted-cyclohexylamino-4-piperidinyl-acetamide antagonists of CCR2

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FIELD OF THE INVENTION The invention is directed to 4-substituted-cyclohexylamino-4-piperidiyl-acetamide compounds, which are antagonists to the chemoattractant cytokine receptor 2 (CCR2), pharmaceutical compositions, and methods for use thereof. Compounds of the invention are useful for preventing,
CROSS REFERENCE TO RELATED APPLICATIONS This application is based on, and claims priority from, provisional application 60/022,056 filed on Jul. 22, 1996. SUMMARY OF THE INVENTION This invention is concerned with a novel process for the synthesis of compounds 9 and 10, both key intermediates in the

Benzoxazepine derivatives and use thereof

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This application is a U.S. national stage of International Application No. PCT/JP2008/054093 filed Mar. 6, 2008. TECHNICAL FIELD The present invention relates to a benzoxazepine derivative having a superior serotonin 5-HT.sub.2C receptor activation action and useful as a drug for the treatment or
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