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Treating androgen decline in aging male (ADAM)-associated conditions with SARMs

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FIELD OF THE INVENTION The present invention relates to a novel class of androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new subclass of compounds, which are selective androgen

Treating androgen decline in aging male (ADAM)-associated conditions with SARMs

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FIELD OF THE INVENTION The present invention relates to a novel class of androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new subclass of compounds, which are selective androgen

Selective androgen receptor modulators

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FIELD OF INVENTION The present invention relates to androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity, which are nonsteroidal ligands for the androgen receptor. The agents are useful for a) male contraception; b) treatment of a variety of hormone-related

Selective androgen receptor modulators

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FIELD OF INVENTION The present invention relates to androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity, which are nonsteroidal ligands for the androgen receptor. The agents are useful for a) male contraception; b) treatment of a variety of hormone-related

Formulations comprising selective androgen receptor modulators

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FIELD OF INVENTION The present invention relates to pharmaceutical compositions and formulations comprising a novel class of androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new

Multi-substituted selective androgen receptor modulators and methods of use thereof

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FIELD OF INVENTION The present invention relates to androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new subclass of compounds, which are selective androgen receptor modulators

Multi-substitued selective androgen receptor modulators and methods of use thereof

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FIELD OF INVENTION The present invention relates to a novel class of androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new subclass of compounds, which are selective androgen receptor

Methylene-bridged selective androgen receptor modulators and methods of use thereof

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FIELD OF INVENTION The present invention relates to a novel class of androgen receptor targeting agents (ARTA), which are selective androgen receptor modulators (SARM). The SARM compounds are useful for a) male contraception; b) treatment of a variety of hormone-related conditions, for example

Heterocyclic selective androgen receptor modulators and methods of use thereof

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FIELD OF INVENTION The present invention relates to a novel class of androgen receptor targeting agents (ARTA), which are selective androgen receptor modulators (SARM). The SARM compounds are useful for a) male contraception; b) treatment of a variety of hormone-related conditions, for example

Halogenated selective androgen receptor modulators and methods of use thereof

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FIELD OF INVENTION The present invention relates to a novel class of androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new subclass of compounds, which are selective androgen receptor

Selective androgen receptor modulators and methods of use thereof

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FIELD OF INVENTION The present invention relates to a novel class of androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new subclass of compounds, which are selective androgen receptor

N-bridged selective androgen receptor modulators and methods of use thereof

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FIELD OF INVENTION The present invention relates to a novel class of androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new subclass of compounds, which are selective androgen receptor

Synthesis of selective androgen receptor modulators

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FIELD OF INVENTION The present invention relates to a synthetic process for the preparation of a novel class of androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new subclass of

Synthesis of selective androgen receptor modulators

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FIELD OF INVENTION The present invention relates to a synthetic process for the preparation of a novel class of androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new subclass of

Methods and compositions for regulation of 5-.alpha.-reductase activity

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TECHNICAL FIELD OF THE INVENTION The present invention relates generally to compounds, compositions methods regulating the action and function of androgens and other steroid hormones by modulating the activity of steroid-reductases, including isozymes of 5.alpha.-reductases. More specifically, the
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