Die Pharmazie 1977-Nov
Penta-acetyl-gitoxin: the prototype of a prodrug in the cardiac glycoside series.
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Penta-acetyl-gitoxin is a suitable prodrug of gitoxin since it shows--side-effect latentiation, due to its inactive application form;--bioavailability, due to its improved solubility and thus good enteral absorption and--bioactivation, due to rapid de-acetylation in the body after absorption.