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Alkanesulfonamido-1-indanone derivatives as inhibitors of cyclooxygenase

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BACKGROUND OF THE INVENTION This invention relates to compounds and pharmaceutical compositions for the treatment of cyclooxygenase mediated diseases and methods of treating thereof. Non-steroidal, antiinflammatory drugs exert most of their antiinflammatory, analgesic and antipyretic activity and

Isoxazolone compounds useful in treating diseases associated with unwanted cytokine activity

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TECHNICAL FIELD The present invention is directed to certain isoxazolone compounds that inhibit the release of inflammatory cytokines such as interleukin-1 (IL-1) and tumor necrosis factor (TNF) from cells. The compounds of the invention, therefore, are useful in treating diseases involving unwanted

Isoxazolone compounds useful in treating diseases associated with unwanted cytokine activity

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Prisijungti Registracija
TECHNICAL FIELD The present invention is directed to certain isoxazolone compounds that inhibit the release of inflammatory cytokines such as interleukin-1 (1L-1) and tumor necrosis factor (TNF) from cells. The compounds of the invention, therefore, are useful in treating diseases involving unwanted
CROSS-REFERENCE TO RELATED APPLICATIONS This application is a 371 of PCT/KR2010/007845, filed Nov. 8, 2010, which claims the benefit of Korean Patent Application No. 10-2009-0106912, filed Nov. 6, 2009, the entire contents of each of which are incorporated herein by reference. TECHNICAL FIELD The

Esters of 3-demethylthiocolchicine and n-acyl analogs

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FIELD OF THE INVENTION The present invention relates to esters of 3-demethylthiocolchicine and N-acyl analogs as substitutes of colchicine in diseases treated with colchicine, particularly liver disorders. Moreover, the invention is concerned with pharmaceutical compositions of the esters of
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