4 полученные результаты
FIELD OF THE INVENTION
This invention relates to derivatives of pentose monosaccharides which exhibit anti-proliferative and anti-inflammatory activity as well as intermediate for the synthesis of these compounds. Compounds of the invention are useful for treating mammals with inflammatory and/or
The present invention relates to galactosylated pro-drugs of non-steroidal anti-inflammatories with free acid function and the process of synthesis thereof, which enables minimization of the gastrointestinal toxicity of the starting anti-inflammatory by means of esterification of its carboxylic
BACKGROUND OF THE INVENTION
Various 2-[(substituted heterocyclic)alkyl]-1H-benz[de]isoquinoline-1,3(2H)-diones having central nervous system and anti-inflammatory activity are disclosed by Wade et al. in U.S. Pat. Nos. 3,935,227; 3,940,397; 3,940,398; 3,947,452; and 3,959,286. Also, Schenker in U.S.
FIELD OF INVENTION
This invention generally relates to the derivatives of 5,6-dideoxy-.alpha.,D-5-epiglucofuranose, 5,6-dideoxy-.alpha.,D-5-epiallofuranose, 5,6-dideoxy-.alpha.,D-5-epimannofuranoside, 5-deoxy-.alpha.,D-lyxofuranoside, 5-deoxy-.alpha.,D-xylofuranose, 5-deoxy-.alpha.,D-ribofuranose,