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ovarian neoplasms/debelost

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13 rezultatov

LKB1-AMPK activators for therapeutic use in polycystic kidney disease

Samo registrirani uporabniki lahko prevajajo članke
Prijava / prijava
BACKGROUND Autosomal dominant polycystic kidney disease (ADPKD) is a frequently inherited kidney disorder with a gene frequency of 1 in 500 to 1,000 births affecting nearly 600,000 Americans and as many as 12 million people worldwide. This potentially lethal genetic disease is characterized by the

Selective androgen receptor modulators

Samo registrirani uporabniki lahko prevajajo članke
Prijava / prijava
FIELD OF INVENTION The present invention relates to androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity, which are nonsteroidal ligands for the androgen receptor. The agents are useful for a) male contraception; b) treatment of a variety of hormone-related

Selective androgen receptor modulators

Samo registrirani uporabniki lahko prevajajo članke
Prijava / prijava
FIELD OF INVENTION The present invention relates to androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity, which are nonsteroidal ligands for the androgen receptor. The agents are useful for a) male contraception; b) treatment of a variety of hormone-related

Formulations comprising selective androgen receptor modulators

Samo registrirani uporabniki lahko prevajajo članke
Prijava / prijava
FIELD OF INVENTION The present invention relates to pharmaceutical compositions and formulations comprising a novel class of androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new

Multi-substituted selective androgen receptor modulators and methods of use thereof

Samo registrirani uporabniki lahko prevajajo članke
Prijava / prijava
FIELD OF INVENTION The present invention relates to androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new subclass of compounds, which are selective androgen receptor modulators

Multi-substitued selective androgen receptor modulators and methods of use thereof

Samo registrirani uporabniki lahko prevajajo članke
Prijava / prijava
FIELD OF INVENTION The present invention relates to a novel class of androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new subclass of compounds, which are selective androgen receptor

Methylene-bridged selective androgen receptor modulators and methods of use thereof

Samo registrirani uporabniki lahko prevajajo članke
Prijava / prijava
FIELD OF INVENTION The present invention relates to a novel class of androgen receptor targeting agents (ARTA), which are selective androgen receptor modulators (SARM). The SARM compounds are useful for a) male contraception; b) treatment of a variety of hormone-related conditions, for example

Heterocyclic selective androgen receptor modulators and methods of use thereof

Samo registrirani uporabniki lahko prevajajo članke
Prijava / prijava
FIELD OF INVENTION The present invention relates to a novel class of androgen receptor targeting agents (ARTA), which are selective androgen receptor modulators (SARM). The SARM compounds are useful for a) male contraception; b) treatment of a variety of hormone-related conditions, for example

Halogenated selective androgen receptor modulators and methods of use thereof

Samo registrirani uporabniki lahko prevajajo članke
Prijava / prijava
FIELD OF INVENTION The present invention relates to a novel class of androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new subclass of compounds, which are selective androgen receptor

Selective androgen receptor modulators and methods of use thereof

Samo registrirani uporabniki lahko prevajajo članke
Prijava / prijava
FIELD OF INVENTION The present invention relates to a novel class of androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new subclass of compounds, which are selective androgen receptor

N-bridged selective androgen receptor modulators and methods of use thereof

Samo registrirani uporabniki lahko prevajajo članke
Prijava / prijava
FIELD OF INVENTION The present invention relates to a novel class of androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new subclass of compounds, which are selective androgen receptor

Synthesis of selective androgen receptor modulators

Samo registrirani uporabniki lahko prevajajo članke
Prijava / prijava
FIELD OF INVENTION The present invention relates to a synthetic process for the preparation of a novel class of androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new subclass of

Synthesis of selective androgen receptor modulators

Samo registrirani uporabniki lahko prevajajo članke
Prijava / prijava
FIELD OF INVENTION The present invention relates to a synthetic process for the preparation of a novel class of androgen receptor targeting agents (ARTA), which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor. The agents define a new subclass of
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