4 rezultatov
BACKGROUND OF THE INVENTION
1. Field of the Invention
The present invention relates to novel compounds, methods, and compositions capable of decreasing HIF hydroxylase enzyme activity, thereby increasing the stability and/or activity of hypoxia inducible factor (HIF).
2. State of the Art
Hypoxia
BACKGROUND OF THE INVENTION
1. Field of the Invention
The present invention relates to novel compounds, methods, and compositions capable of decreasing HIF hydroxylase enzyme activity, thereby increasing the stability and/or activity of hypoxia inducible factor (HIF).
2. State of the Art
Hypoxia
BACKGROUND OF THE INVENTION
1. Field of the Invention
The present invention relates to novel compounds capable of modulating the stability and/or activity of hypoxia inducible factor (HIF).
2. State of the Art
Hypoxia inducible factor (HIF) is a basic helix-loop-helix (bHLH) PAS (Per/Arnt/Sim)
FEATURES OF THE INVENTION
The present invention relates to novel dibenz[b,e]oxepin derivatives useful for prevention and treatment of cerebral diseases caused by hypoxia.
TECHNICAL BACKGROUND
The brain, different from other organs, exists under particular environment such that it is dipped in